Primary Site >> Colorectal Cancer

Gene >> PDE5A

Journal: Cancer Res. 2000 Jul 1;60(13):3338-42.
Title: Exisulind induction of apoptosis involves guanosine 3',5'-cyclic monophosphate phosphodiesterase inhibition, protein kinase G activation, and attenuated beta-catenin.
Author: Thompson, W J|Piazza, G A|Li, H|Liu, L|Fetter, J|Zhu, B|Sperl, G|Ahnen, D|Pamukcu, R
PMID: 10910034
Journal: Cancer Res. 2001 May 15;61(10):3961-8.
Title: Exisulind, a novel proapoptotic drug, inhibits rat urinary bladder tumorigenesis.
Author: Piazza, G A|Thompson, W J|Pamukcu, R|Alila, H W|Whitehead, C M|Liu, L|Fetter, J R|Gresh, W E Jr|Klein-Szanto, A J|Farnell, D R|Eto, I|Grubbs, C J
PMID: 11358813
Journal: Cell Signal. 2002 Jan;14(1):45-51.
Title: Specific cGMP binding by the cGMP binding domains of cGMP-binding cGMP specific phosphodiesterase.
Author: Liu, Li|Underwood, Tashandra|Li, Han|Pamukcu, Rifat|Thompson, W Joseph
PMID: 11747988
Journal: J Cell Biochem. 2005 Feb 1;94(2):336-50.
Title: Suppression of cyclic GMP-specific phosphodiesterase 5 promotes apoptosis and inhibits growth in HT29 cells.
Author: Zhu, Bing|Vemavarapu, Lakshmi|Thompson, W Joseph|Strada, Samuel J
PMID: 15526282
Journal: Int J Oncol. 2008 May;32(5):975-83.
Title: Characterization of gene expression regulated by American ginseng and ginsenoside Rg3 in human colorectal cancer cells.
Author: Luo, Xiaoji|Wang, Chong-Zhi|Chen, Jin|Song, Wen-Xin|Luo, Jinyong|Tang, Ni|He, Bai-Cheng|Kang, Quan|Wang, Yitao|Du, Wei|He, Tong-Chuan|Yuan, Chun-Su
PMID: 18425323
Journal: Arzneimittelforschung. 2009;59(8):415-21.
Title: Synthesis of novel tadalafil analogues and their evaluation as phosphodiesterase inhibitors and anticancer agents.
Author: Abadi, Ashraf H|Abouel-Ella, Dalal A|Ahmed, Nermin S|Gary, Bernard D|Thaiparambil, Jose T|Tinsley, Heather N|Keeton, Adam B|Piazza, Gary A
PMID: 19813465
Journal: Eur J Med Chem. 2010 Apr;45(4):1278-86.
Title: Synthesis, molecular modeling and biological evaluation of novel tadalafil analogues as phosphodiesterase 5 and colon tumor cell growth inhibitors, new stereochemical perspective.
Author: Abadi, Ashraf H|Gary, Bernard D|Tinsley, Heather N|Piazza, Gary A|Abdel-Halim, Mohammad
PMID: 20206015
Journal: Cancer Prev Res (Phila). 2010 Oct;3(10):1303-13.
Title: Colon tumor cell growth-inhibitory activity of sulindac sulfide and other nonsteroidal anti-inflammatory drugs is associated with phosphodiesterase 5 inhibition.
Author: Tinsley, Heather N|Gary, Bernard D|Thaiparambil, Jose|Li, Nan|Lu, Wenyan|Li, Yonghe|Maxuitenko, Yulia Y|Keeton, Adam B|Piazza, Gary A
PMID: 20876730
Journal: Cancer Prev Res (Phila). 2012 Jun;5(6):822-33.
Title: A novel sulindac derivative that potently suppresses colon tumor cell growth by inhibiting cGMP phosphodiesterase and beta-catenin transcriptional activity.
Author: Whitt, Jason D|Li, Nan|Tinsley, Heather N|Chen, Xi|Zhang, Wei|Li, Yonghe|Gary, Bernard D|Keeton, Adam B|Xi, Yaguang|Abadi, Ashraf H|Grizzle, William E|Piazza, Gary A
PMID: 22556201
Journal: Mol Cancer Ther. 2013 Sep;12(9):1848-59.
Title: Sulindac selectively inhibits colon tumor cell growth by activating the cGMP/PKG pathway to suppress Wnt/beta-catenin signaling.
Author: Li, Nan|Xi, Yaguang|Tinsley, Heather N|Gurpinar, Evrim|Gary, Bernard D|Zhu, Bing|Li, Yonghe|Chen, Xi|Keeton, Adam B|Abadi, Ashraf H|Moyer, Mary P|Grizzle, William E|Chang, Wen-Chi|Clapper, Margie L|Piazza, Gary A
PMID: 23804703
Journal: J Clin Invest. 2013 Feb;123(2):787-99.
Title: 67-kDa laminin receptor increases cGMP to induce cancer-selective apoptosis.
Author: Kumazoe, Motofumi|Sugihara, Kaori|Tsukamoto, Shuntaro|Huang, Yuhui|Tsurudome, Yukari|Suzuki, Takashi|Suemasu, Yumi|Ueda, Naoki|Yamashita, Shuya|Kim, Yoonhee|Yamada, Koji|Tachibana, Hirofumi
PMID: 23348740
Journal: J Cell Physiol. 2015 Sep;230(9):2281-98.
Title: Nexavar/Stivarga and viagra interact to kill tumor cells.
Author: Tavallai, Mehrad|Hamed, Hossein A|Roberts, Jane L|Cruickshanks, Nichola|Chuckalovcak, John|Poklepovic, Andrew|Booth, Laurence|Dent, Paul
PMID: 25704960
Journal: Oncotarget. 2015 Sep 29;6(29):27403-15.
Title: Suppression of beta-catenin/TCF transcriptional activity and colon tumor cell growth by dual inhibition of PDE5 and 10.
Author: Li, Nan|Chen, Xi|Zhu, Bing|Ramirez-Alcantara, Veronica|Canzoneri, Joshua C|Lee, Kevin|Sigler, Sara|Gary, Bernard|Li, Yonghe|Zhang, Wei|Moyer, Mary P|Salter, E Alan|Wierzbicki, Andrzej|Keeton, Adam B|Piazza, Gary A
PMID: 26299804
Journal: Am J Cancer Res. 2015 Oct 15;5(11):3311-24. eCollection 2015.
Title: Sildenafil inhibits the growth of human colorectal cancer in vitro and in vivo.
Author: Mei, Xiao-Long|Yang, Yang|Zhang, Yao-Jun|Li, Yong|Zhao, Jin-Ming|Qiu, Jian-Ge|Zhang, Wen-Ji|Jiang, Qi-Wei|Xue, You-Qiu|Zheng, Di-Wei|Chen, Yao|Qin, Wu-Ming|Wei, Meng-Ning|Shi, Zhi
PMID: 26807313
Journal: PLoS Med. 2016 Jun 14;13(6):e1002037.
Title: Phosphodiesterase Type 5 Inhibitors and Risk of Malignant Melanoma: Matched Cohort Study Using Primary Care Data from the UK Clinical Practice Research Datalink.
Author: Matthews, Anthony|Langan, Sinead M|Douglas, Ian J|Smeeth, Liam|Bhaskaran, Krishnan
PMID: 27299522
Journal: BMC Cancer. 2016 Dec 7;16(1):938.
Title: Phosphodiesterases in non-neoplastic appearing colonic mucosa from patients with colorectal neoplasia.
Author: Mahmood, Badar|Damm, Morten Matthiesen Bach|Jensen, Thorbjorn Soren Ronn|Backe, Marie Balslev|Dahllof, Mattias Salling|Poulsen, Steen Seier|Bindslev, Niels|Hansen, Mark Berner
PMID: 27927168
Journal: Cancer Prev Res (Phila). 2017 Jul;10(7):377-388.
Title: Sildenafil Suppresses Inflammation-Driven Colorectal Cancer in Mice.
Author: Islam, Bianca N|Sharman, Sarah K|Hou, Yali|Bridges, Allison E|Singh, Nagendra|Kim, Sangmi|Kolhe, Ravindra|Trillo-Tinoco, Jimena|Rodriguez, Paulo C|Berger, Franklin G|Sridhar, Subbaramiah|Browning, Darren D
PMID: 28468928
Journal: Oncotarget. 2017 Aug 2;8(59):99451-99469.
Title: Curcumin interacts with sildenafil to kill GI tumor cells via endoplasmic reticulum stress and reactive oxygen/ nitrogen species.
Author: Roberts, Jane L|Poklepovic, Andrew|Booth, Laurence
PMID: 29245915
Journal: Cancer Prev Res (Phila). 2018 Feb;11(2):81-92.
Title: Cyclic-GMP-Elevating Agents Suppress Polyposis in Apc(Min) mice by Targeting the Preneoplastic Epithelium.
Author: Sharman, Sarah K|Islam, Bianca N|Hou, Yali|Singh, Nagendra|Berger, Franklin G|Sridhar, Subbaramiah|Yoo, Wonsuk|Browning, Darren D
PMID: 29301746
Journal: Cancer Prev Res (Phila). 2018 Jul;11(7):439-440.
Title: Mutations of the PDE5A Gene Confer a Survival Advantage in Patients with Colon Cancer.
Author: Lehrer, Steven|Rheinstein, Peter H|Rosenzweig, Kenneth E
PMID: 29724712
Journal: Semin Cancer Biol. 2018 Sep 3. pii: S1044-579X(18)30064-6.
Title: Targeting the paracrine hormone-dependent guanylate cyclase/cGMP/phosphodiesterases signaling pathway for colorectal cancer prevention.
Author: Yarla, N S|Gali, H|Pathuri, G|Smriti, S|Farooqui, M|Panneerselvam, J|Kumar, G|Madka, V|Rao, C V
PMID: 30189250