Primary Site >> Colorectal Cancer

Gene >> PDE4A

Journal: Cancer Res. 2001 May 15;61(10):3961-8.
Title: Exisulind, a novel proapoptotic drug, inhibits rat urinary bladder tumorigenesis.
Author: Piazza, G A|Thompson, W J|Pamukcu, R|Alila, H W|Whitehead, C M|Liu, L|Fetter, J R|Gresh, W E Jr|Klein-Szanto, A J|Farnell, D R|Eto, I|Grubbs, C J
PMID: 11358813
Journal: Cancer Res. 2007 Jun 1;67(11):5248-57.
Title: Chemoresistant KM12C colon cancer cells are addicted to low cyclic AMP levels in a phosphodiesterase 4-regulated compartment via effects on phosphoinositide 3-kinase.
Author: McEwan, David G|Brunton, Valerie G|Baillie, George S|Leslie, Nicholas R|Houslay, Miles D|Frame, Margaret C
PMID: 17545604
Journal: Mol Cancer. 2012 Jul 25;11:46.
Title: Inhibition of phosphodiesterase-4 (PDE4) activity triggers luminal apoptosis and AKT dephosphorylation in a 3-D colonic-crypt model.
Author: Tsunoda, Toshiyuki|Ota, Takeharu|Fujimoto, Takahiro|Doi, Keiko|Tanaka, Yoko|Yoshida, Yasuhiro|Ogawa, Masahiro|Matsuzaki, Hiroshi|Hamabashiri, Masato|Tyson, Darren R|Kuroki, Masahide|Miyamoto, Shingo|Shirasawa, Senji
PMID: 22830422
Journal: Bioorg Med Chem Lett. 2013 Dec 15;23(24):6721-7.
Title: Synthesis and biological evaluation of nimesulide based new class of triazole derivatives as potential PDE4B inhibitors against cancer cells.
Author: Mareddy, Jyoti|Nallapati, Suresh Babu|Anireddy, Jayasree|Devi, Yumnam Priyadarshini|Mangamoori, Lakshmi Narasu|Kapavarapu, Ravikumar|Pal, Sarbani
PMID: 24215890
Journal: Arch Pharm (Weinheim). 2014 Sep;347(9):650-7.
Title: Novel quinazolin-4(3H)-one/Schiff base hybrids as antiproliferative and phosphodiesterase 4 inhibitors: design, synthesis, and docking studies.
Author: Abdel-Rahman, Hamdy M|Abdel-Aziz, Mohamed|Canzoneri, Joshua C|Gary, Bernard D|Piazza, Gary A
PMID: 24985336
Journal: Anticancer Res. 2014 Aug;34(8):4551-5.
Title: Resveratrol induces luminal apoptosis of human colorectal cancer HCT116 cells in three-dimensional culture.
Author: Tsunoda, Toshiyuki|Ishikura, Shuhei|Doi, Keiko|Matsuzaki, Hiroshi|Iwaihara, Yuri|Shirasawa, Senji
PMID: 25075098
Journal: BMC Cancer. 2016 Dec 7;16(1):938.
Title: Phosphodiesterases in non-neoplastic appearing colonic mucosa from patients with colorectal neoplasia.
Author: Mahmood, Badar|Damm, Morten Matthiesen Bach|Jensen, Thorbjorn Soren Ronn|Backe, Marie Balslev|Dahllof, Mattias Salling|Poulsen, Steen Seier|Bindslev, Niels|Hansen, Mark Berner
PMID: 27927168
Journal: Int Immunopharmacol. 2018 Mar;56:36-42.
Title: Roflumilast, type 4 phosphodiesterase inhibitor, attenuates inflammation in rats with ulcerative colitis via down-regulation of iNOS and elevation of cAMP.
Author: El-Ashmawy, Nahla E|Khedr, Naglaa F|El-Bahrawy, Hoda A|El-Adawy, Samar A
PMID: 29331766