Primary Site >> Colorectal Cancer

Gene >> NEDD8

Journal: Hepatology. 2012 Apr;55(4):1237-48.
Title: Murine double minute 2 regulates Hu antigen R stability in human liver and colon cancer through NEDDylation.
Author: Embade, Nieves|Fernandez-Ramos, David|Varela-Rey, Marta|Beraza, Naiara|Sini, Marcella|Gutierrez de Juan, Virginia|Woodhoo, Ashwin|Martinez-Lopez, Nuria|Rodriguez-Iruretagoyena, Begona|Bustamante, Francisco Javier|de la Hoz, Ana Belen|Carracedo, Arkaitz|Xi
PMID: 22095636
Journal: Cell Rep. 2012 Apr 19;1(4):309-16.
Title: A gatekeeper residue for NEDD8-activating enzyme inhibition by MLN4924.
Author: Toth, Julia I|Yang, Li|Dahl, Russell|Petroski, Matthew D
PMID: 22832224
Journal: Cancer Res. 2013 Jan 1;73(1):225-34.
Title: Novel DNA damage checkpoints mediating cell death induced by the NEDD8-activating enzyme inhibitor MLN4924.
Author: Blank, Jonathan L|Liu, Xiaozhen J|Cosmopoulos, Katherine|Bouck, David C|Garcia, Khristofer|Bernard, Hugues|Tayber, Olga|Hather, Greg|Liu, Ray|Narayanan, Usha|Milhollen, Michael A|Lightcap, Eric S
PMID: 23100467
Journal: Nat Commun. 2014 May 13;5:3733.
Title: The covalent modifier Nedd8 is critical for the activation of Smurf1 ubiquitin ligase in tumorigenesis.
Author: Xie, Ping|Zhang, Minghua|He, Shan|Lu, Kefeng|Chen, Yuhan|Xing, Guichun|Lu, Yiming|Liu, Ping|Li, Yang|Wang, Shaoxia|Chai, Nan|Wu, Jiawei|Deng, Haiteng|Wang, Hong-Rui|Cao, Yu|Zhao, Fei|Cui, Yu|Wang, Jian|He, Fuchu|Zhang, Lingqiang
PMID: 24821572
Journal: Am J Cancer Res. 2015 Oct 15;5(11):3400-6. eCollection 2015.
Title: Molecular dynamics simulation on the low sensitivity of mutants of NEDD-8 activating enzyme for MLN4924 inhibitor as a cancer drug.
Author: Rashidieh, Behnam|Valizadeh, Mohharam|Assadollahi, Vahideh|Ranjbar, Mohammad Mehdi
PMID: 26807320
Journal: Technol Cancer Res Treat. 2016 Aug;15(4):527-34.
Title: Radiosensitization of Human Colorectal Cancer Cells by MLN4924: An Inhibitor of NEDD8-Activating Enzyme.
Author: Wan, Juefeng|Zhu, Ji|Li, Guichao|Zhang, Zhen
PMID: 26082455
Journal: J Natl Cancer Inst. 2016 Oct 22;109(2). pii: djw209.
Title: Efficacy of NEDD8 Pathway Inhibition in Preclinical Models of Poorly Differentiated, Clinically Aggressive Colorectal Cancer.
Author: Picco, Gabriele|Petti, Consalvo|Sassi, Francesco|Grillone, Katia|Migliardi, Giorgia|Rossi, Teresa|Isella, Claudio|Di Nicolantonio, Federica|Sarotto, Ivana|Sapino, Anna|Bardelli, Alberto|Trusolino, Livio|Bertotti, Andrea|Medico, Enzo
PMID: 27771609
Journal: Eur J Med Chem. 2017 Jun 16;133:174-183.
Title: Discovery of benzothiazole derivatives as novel non-sulfamide NEDD8 activating enzyme inhibitors by target-based virtual screening.
Author: Ma, Hao|Zhuang, Chunlin|Xu, Xiguo|Li, Jiao|Wang, Juan|Min, Xiao|Zhang, Wannian|Zhang, Huojun|Miao, Zhenyuan
PMID: 28388520
Journal: Mol Med Rep. 2017 May;15(5):2795-2801.
Title: Neural precursor cell expressed, developmentally downregulated 8activating enzyme inhibitor MLN4924 sensitizes colorectal cancer cells to oxaliplatin by inducing DNA damage, G2 cell cycle arrest and apoptosis.
Author: Zheng, Wanwei|Luo, Zhongguang|Zhang, Jun|Min, Pei|Li, Wenshuai|Xu, Diannan|Zhang, Ziqiang|Xiong, Panpan|Liang, Hong|Liu, Jie
PMID: 28447739
Journal: Anticancer Drugs. 2018 Oct;29(9):854-860.
Title: Construction and characterization of regulated cycle inhibiting factors induced upon Tet-On system in human colon cancer cell lines.
Author: Liu, Liang|Ni, Jianjiao|Zhang, Junhua|He, Xinhong
PMID: 29923895