Primary Site >> Colorectal Cancer

Gene >> CES2

Journal: Clin Cancer Res. 2002 Aug;8(8):2605-11.
Title: Human carboxylesterase 2 is commonly expressed in tumor tissue and is correlated with activation of irinotecan.
Author: Xu, Guang|Zhang, Wanghai|Ma, Margaret K|McLeod, Howard L
PMID: 12171891
Journal: Br J Cancer. 2002 Sep 9;87(6):659-64.
Title: Secreted and tumour targeted human carboxylesterase for activation of irinotecan.
Author: Oosterhoff, D|Pinedo, H M|van der Meulen, I H|de Graaf, M|Sone, T|Kruyt, F A|van Beusechem, V W|Haisma, H J|Gerritsen, W R
PMID: 12237777
Journal: Cancer Chemother Pharmacol. 2002 Apr;49(4):329-35.
Title: Determinants of the cytotoxicity of irinotecan in two human colorectal tumor cell lines.
Author: Pavillard, Valerie|Agostini, Cecile|Richard, Sophie|Charasson, Virginie|Montaudon, Daniele|Robert, Jacques
PMID: 11914913
Journal: Clin Cancer Res. 2003 Oct 15;9(13):4983-91.
Title: Carboxylesterases expressed in human colon tumor tissue and their role in CPT-11 hydrolysis.
Author: Sanghani, Sonal P|Quinney, Sara K|Fredenburg, Tyler B|Sun, Zejin|Davis, Wilhelmina I|Murry, Daryl J|Cummings, Oscar W|Seitz, David E|Bosron, William F
PMID: 14581373
Journal: Br J Cancer. 2005 Jan 31;92(2):259-64.
Title: Unfavourable expression of pharmacologic markers in mucinous colorectal cancer.
Author: Glasgow, S C|Yu, J|Carvalho, L P|Shannon, W D|Fleshman, J W|McLeod, H L
PMID: 15655543
Journal: J Pharmacol Exp Ther. 2005 Jun;313(3):1011-6.
Title: Hydrolysis of capecitabine to 5'-deoxy-5-fluorocytidine by human carboxylesterases and inhibition by loperamide.
Author: Quinney, S K|Sanghani, S P|Davis, W I|Hurley, T D|Sun, Z|Murry, D J|Bosron, W F
PMID: 15687373
Journal: Clin Cancer Res. 2005 Oct 1;11(19 Pt 1):6901-7.
Title: Carboxylesterase isoform 2 mRNA expression in peripheral blood mononuclear cells is a predictive marker of the irinotecan to SN38 activation step in colorectal cancer patients.
Author: Cecchin, Erika|Corona, Giuseppe|Masier, Sara|Biason, Paola|Cattarossi, Giulio|Frustaci, Sergio|Buonadonna, Angela|Colussi, Annamaria|Toffoli, Giuseppe
PMID: 16203781
Journal: Cancer Biol Ther. 2006 Nov;5(11):1450-6. Epub 2006 Nov 13.
Title: Transcriptional activation of the carboxylesterase 2 gene by the p53 pathway.
Author: Choi, Woonyoung|Cogdell, David|Feng, Yumei|Hamilton, Stanley R|Zhang, Wei
PMID: 16963839
Journal: J Pharmacol Exp Ther. 2007 Oct;323(1):94-101.
Title: Expression and characterization of a human carboxylesterase 2 splice variant.
Author: Schiel, Marissa A|Green, Scheri-lyn|Davis, Wilhelmina I|Sanghani, Paresh C|Bosron, William F|Sanghani, Sonal P
PMID: 17636009
Journal: Cancer Chemother Pharmacol. 2008 Mar;61(3):481-8. Epub 2007 May 5.
Title: Functional study of the 830C>G polymorphism of the human carboxylesterase 2 gene.
Author: Bellott, Ricardo|Le Morvan, Valerie|Charasson, Virginie|Laurand, Armelle|Colotte, Marthe|Zanger, Ulrich M|Klein, Kathrin|Smith, Denis|Bonnet, Jacques|Robert, Jacques
PMID: 17483951
Journal: Cancer Invest. 2008 Mar;26(2):178-81.
Title: Carboxylesterase 2 is downregulated in colorectal cancer following progression of the disease.
Author: Tang, Xiaobo|Wu, Hong|Wu, Zhenghua|Wang, Guiyu|Wang, Zhigang|Zhu, Daling
PMID: 18259949
Journal: Curr Drug Metab. 2008 May;9(4):336-43.
Title: A carboxylesterase 2 gene polymorphism as predictor of capecitabine on response and time to progression.
Author: Ribelles, N|Lopez-Siles, J|Sanchez, A|Gonzalez, E|Sanchez, M J|Carabantes, F|Sanchez-Rovira, P|Marquez, A|Duenas, R|Sevilla, I|Alba, E
PMID: 18473752
Journal: Br J Cancer. 2008 Oct 21;99(8):1239-45.
Title: Pharmacokinetic and pharmacogenetic determinants of the activity and toxicity of irinotecan in metastatic colorectal cancer patients.
Author: Rouits, E|Charasson, V|Petain, A|Boisdron-Celle, M|Delord, J-P|Fonck, M|Laurand, A|Poirier, A-L|Morel, A|Chatelut, E|Robert, J|Gamelin, E
PMID: 18797458
Journal: Drug Metab Dispos. 2009 Jul;37(7):1539-47.
Title: Regulation of tissue-specific carboxylesterase expression by pregnane x receptor and constitutive androstane receptor.
Author: Xu, Chenshu|Wang, Xinkun|Staudinger, Jeff L
PMID: 19359405
Journal: Tumori. 2009 Jul-Aug;95(4):473-8.
Title: Decreased serum levels of carboxylesterase-2 in patients with ovarian cancer.
Author: Cai, Liying|Tang, Xiaobo|Guo, Lei|An, Yuan|Wang, Yuguang|Zheng, Jianhua
PMID: 19856659
Journal: Int J Cancer. 2010 Sep 1;127(5):1028-37.
Title: Evidence of heterogeneity within colorectal liver metastases for allelic losses, mRNA level expression and in vitro response to chemotherapeutic agents.
Author: Goasguen, Nicolas|de Chaisemartin, Cecile|Brouquet, Antoine|Julie, Catherine|Prevost, Gregoire P|Laurent-Puig, Pierre|Penna, Christophe
PMID: 20017140
Journal: Clin Cancer Res. 2011 Apr 1;17(7):2006-13.
Title: A polymorphism in the cytidine deaminase promoter predicts severe capecitabine-induced hand-foot syndrome.
Author: Caronia, Daniela|Martin, Miguel|Sastre, Javier|de la Torre, Julio|Garcia-Saenz, Jose Angel|Alonso, Maria R|Moreno, Leticia T|Pita, Guillermo|Diaz-Rubio, Eduardo|Benitez, Javier|Gonzalez-Neira, Anna
PMID: 21325291
Journal: PLoS Comput Biol. 2011 Sep;7(9):e1002143.
Title: A combined experimental and mathematical approach for molecular-based optimization of irinotecan circadian delivery.
Author: Ballesta, Annabelle|Dulong, Sandrine|Abbara, Chadi|Cohen, Boris|Okyar, Alper|Clairambault, Jean|Levi, Francis
PMID: 21931543
Journal: Cancer Chemother Pharmacol. 2012 Jul;70(1):25-32.
Title: Phase II and gene expression analysis trial of neoadjuvant capecitabine plus irinotecan followed by capecitabine-based chemoradiotherapy for locally advanced rectal cancer: Hoosier Oncology Group GI03-53.
Author: Chiorean, E Gabriela|Sanghani, Sonal|Schiel, Marissa A|Yu, Menggang|Burns, Matthew|Tong, Yan|Hinkle, David T|Coleman, Nicki|Robb, Bruce|LeBlanc, Julia|Clark, Romnee|Bufill, Jose|Curie, Colleen|Loehrer, Patrick J|Cardenes, Higinia
PMID: 22610353
Journal: Br J Pharmacol. 2013 Apr;168(8):1989-99.
Title: Regulation of carboxylesterase-2 expression by p53 family proteins and enhanced anti-cancer activities among 5-fluorouracil, irinotecan and doxazolidine prodrug.
Author: Xiao, Da|Yang, Dongfang|Guo, Liangran|Lu, Wei|Charpentier, Margaret|Yan, Bingfang
PMID: 23373735
Journal: Neoplasma. 2014;61(1):99-109.
Title: Relationship between the expression of CES2, UGT1A1, and GUSB in colorectal cancer tissues and aberrant methylation.
Author: Xie, F W|Peng, Y|Chen, Xiong|Chen, Xi|Li, J|Wang, W|Yu, Z|Ouyang, X
PMID: 24195516
Journal: Biomed Pharmacother. 2014 Feb;68(1):31-7.
Title: Regulation and expression of aberrant methylation on irinotecan metabolic genes CES2, UGT1A1 and GUSB in the in-vitro cultured colorectal cancer cells.
Author: Xie, Fang-Wei|Peng, Yong-Hai|Chen, Xi|Chen, Xiong|Li, Jie|Yu, Zong-Yang|Wang, Wen-Wu|Ouyang, Xue-Nong
PMID: 24439671
Journal: J Pharmacol Exp Ther. 2014 Oct;351(1):61-6.
Title: Pegylation improves the pharmacokinetics and bioavailability of small-molecule drugs hydrolyzable by esterases: a study of phospho-Ibuprofen.
Author: Mattheolabakis, George|Wong, Chi C|Sun, Yu|Amella, Carol A|Richards, Robert|Constantinides, Panayiotis P|Rigas, Basil
PMID: 25047517
Journal: Int J Mol Sci. 2014 Sep 5;15(9):15767-77.
Title: CES2, ABCG2, TS and Topo-I primary and synchronous metastasis expression and clinical outcome in metastatic colorectal cancer patients treated with first-line FOLFIRI regimen.
Author: Silvestris, Nicola|Simone, Giovanni|Partipilo, Giulia|Scarpi, Emanuela|Lorusso, Vito|Brunetti, Anna Elisabetta|Maiello, Evaristo|Paradiso, Angelo|Mangia, Anita
PMID: 25198900
Journal: Biomed Pharmacother. 2014 Sep;68(7):825-31.
Title: Influence of UGT1A1 gene methylation level in colorectal cancer cells on the sensitivity of the chemotherapy drug CPT-11.
Author: Xie, Fang-Wei|Peng, Yong-Hai|Wang, Wen-Wu|Chen, Xi|Chen, Xiong|Li, Jie|Yu, Zong-Yang|Ouyang, Xue-Nong
PMID: 25260839
Journal: Cancer Lett. 2016 Aug 1;378(1):51-8.
Title: Tissue-infiltrating plasma cells are an important source of carboxylesterase 2 contributing to the therapeutic efficacy of prodrugs.
Author: Kuhl, Anja A|Erben, Ulrike|Cieluch, Constanze|Spieckermann, Simone|Grone, Jorn|Lohneis, Philipp|Pape, Ulrich Frank|Arsenic, Ruza|Utku, Nalan
PMID: 27149931
Journal: Oncotarget. 2016 Nov 15;7(46):75279-75292.
Title: High-throughput proteomics integrated with gene microarray for discovery of colorectal cancer potential biomarkers.
Author: Yu, Jiekai|Li, Xiaofen|Zhong, Chenhan|Li, Dan|Zhai, Xiaohui|Hu, Wangxiong|Guo, Cheng|Yuan, Ying|Zheng, Shu
PMID: 27661117
Journal: Chembiochem. 2017 Jul 4;18(13):1204-1215.
Title: Glycoengineering of Esterase Activity through Metabolic Flux-Based Modulation of Sialic Acid.
Author: Mathew, Mohit P|Tan, Elaine|Labonte, Jason W|Shah, Shivam|Saeui, Christopher T|Liu, Lingshu|Bhattacharya, Rahul|Bovonratwet, Patawut|Gray, Jeffrey J|Yarema, Kevin J
PMID: 28218815
Journal: Dis Markers. 2018 Jan 31;2018:5280736.
Title: The Relationship between TP53 Gene Status and Carboxylesterase 2 Expression in Human Colorectal Cancer.
Author: Ishimine, Momoko|Lee, Hyeon-Cheol|Nakaoka, Hirofumi|Orita, Hajime|Kobayashi, Toshiyuki|Mizuguchi, Konomi|Endo, Mikumi|Inoue, Ituro|Sato, Koichi|Yokomizo, Takehiko
PMID: 29651325
Journal: Biol Pharm Bull. 2018;41(5):697-706.
Title: Development of a Caco-2 Cell Line Carrying the Human Intestine-Type CES Expression Profile as a Promising Tool for Ester-Containing Drug Permeability Studies.
Author: Ishizaki, Yuma|Furihata, Tomomi|Oyama, Yusuke|Ohura, Kayoko|Imai, Teruko|Hosokawa, Masakiyo|Akita, Hidetaka|Chiba, Kan
PMID: 29709907