Primary Site >> Colorectal Cancer

Gene >> CDK19

Journal: Mol Carcinog. 2013 Jun;52(6):459-74.
Title: Histone deacetylase inhibition in colorectal cancer cells reveals competing roles for members of the oncogenic miR-17-92 cluster.
Author: Humphreys, Karen J|Cobiac, Lynne|Le Leu, Richard K|Van der Hoek, Mark B|Michael, Michael Z
PMID: 22308110
Journal: J Med Chem. 2016 Feb 11;59(3):1078-101.
Title: Discovery of Potent, Selective, and Orally Bioavailable Small-Molecule Modulators of the Mediator Complex-Associated Kinases CDK8 and CDK19.
Author: Mallinger, Aurelie|Schiemann, Kai|Rink, Christian|Stieber, Frank|Calderini, Michel|Crumpler, Simon|Stubbs, Mark|Adeniji-Popoola, Olajumoke|Poeschke, Oliver|Busch, Michael|Czodrowski, Paul|Musil, Djordje|Schwarz, Daniel|Ortiz-Ruiz, Maria-Jesus|Schneider, R
PMID: 26796641
Journal: Bioorg Med Chem Lett. 2016 Mar 1;26(5):1443-51.
Title: Discovery of potent and selective CDK8 inhibitors from an HSP90 pharmacophore.
Author: Schiemann, Kai|Mallinger, Aurelie|Wienke, Dirk|Esdar, Christina|Poeschke, Oliver|Busch, Michael|Rohdich, Felix|Eccles, Suzanne A|Schneider, Richard|Raynaud, Florence I|Czodrowski, Paul|Musil, Djordje|Schwarz, Daniel|Urbahns, Klaus|Blagg, Julian
PMID: 26852363
Journal: Front Pharmacol. 2017 Feb 2;8:38.
Title: Pharmacogenomic Characterization and Isobologram Analysis of the Combination of Ascorbic Acid and Curcumin-Two Main Metabolites of Curcuma longa-in Cancer Cells.
Author: Ooko, Edna|Kadioglu, Onat|Greten, Henry J|Efferth, Thomas
PMID: 28210221
Journal: Cell Rep. 2017 Nov 7;21(6):1495-1506.
Title: CDK8 Kinase Activity Promotes Glycolysis.
Author: Galbraith, Matthew D|Andrysik, Zdenek|Pandey, Ahwan|Hoh, Maria|Bonner, Elizabeth A|Hill, Amanda A|Sullivan, Kelly D|Espinosa, Joaquin M
PMID: 29117556
Journal: J Biol Chem. 2018 Mar 30;293(13):4870-4882.
Title: Oncogenic exon 2 mutations in Mediator subunit MED12 disrupt allosteric activation of cyclin C-CDK8/19.
Author: Park, Min Ju|Shen, Hailian|Spaeth, Jason M|Tolvanen, Jaana H|Failor, Courtney|Knudtson, Jennifer F|McLaughlin, Jessica|Halder, Sunil K|Yang, Qiwei|Bulun, Serdar E|Al-Hendy, Ayman|Schenken, Robert S|Aaltonen, Lauri A|Boyer, Thomas G
PMID: 29440396
Journal: Mol Cell Biol. 2018 May 15;38(11). pii: MCB.00573-17.
Title: Depletion of Mediator Kinase Module Subunits Represses Superenhancer-Associated Genes in Colon Cancer Cells.
Author: Kuuluvainen, Emilia|Domenech-Moreno, Eva|Niemela, Elina H|Makela, Tomi P
PMID: 29507187