Primary Site >> Pancreatic Cancer

Gene >> BRD4

Journal: Mol Cancer Ther. 2014 Jul;13(7):1907-17.
Title: BET bromodomain inhibitors block growth of pancreatic cancer cells in three-dimensional collagen.
Author: Sahai, Vaibhav|Kumar, Krishan|Knab, Lawrence M|Chow, Christina R|Raza, Sania S|Bentrem, David J|Ebine, Kazumi|Munshi, Hidayatullah G
PMID: 24807963
Journal: Sci Rep. 2015 Mar 25;5:9489.
Title: GLI2-dependent c-MYC upregulation mediates resistance of pancreatic cancer cells to the BET bromodomain inhibitor JQ1.
Author: Kumar, Krishan|Raza, Sania S|Knab, Lawrence M|Chow, Christina R|Kwok, Benjamin|Bentrem, David J|Popovic, Relja|Ebine, Kazumi|Licht, Jonathan D|Munshi, Hidayatullah G
PMID: 25807524
Journal: Oncotarget. 2016 Nov 15;7(46):74415-74426.
Title: Characterization of pancreatic glucagon-producing tumors and pituitary gland tumors in transgenic mice overexpressing MYCN in hGFAP-positive cells.
Author: Fielitz, Kathrin|Althoff, Kristina|De Preter, Katleen|Nonnekens, Julie|Ohli, Jasmin|Elges, Sandra|Hartmann, Wolfgang|Kloppel, Gunter|Knosel, Thomas|Schulte, Marc|Klein-Hitpass, Ludger|Beisser, Daniela|Reis, Henning|Eyking, Annette|Cario, Elke|Schulte, Joh
PMID: 27769070
Journal: JCI Insight. 2017 Feb 9;2(3):e88032.
Title: BET inhibitors block pancreatic stellate cell collagen I production and attenuate fibrosis in vivo.
Author: Kumar, Krishan|DeCant, Brian T|Grippo, Paul J|Hwang, Rosa F|Bentrem, David J|Ebine, Kazumi|Munshi, Hidayatullah G
PMID: 28194432
Journal: Nucleic Acids Res. 2017 Jun 20;45(11):6334-6349.
Title: Histone deacetylase class-I inhibition promotes epithelial gene expression in pancreatic cancer cells in a BRD4- and MYC-dependent manner.
Author: Mishra, Vivek Kumar|Wegwitz, Florian|Kosinsky, Robyn Laura|Sen, Madhobi|Baumgartner, Roland|Wulff, Tanja|Siveke, Jens T|Schildhaus, Hans-Ulrich|Najafova, Zeynab|Kari, Vijayalakshmi|Kohlhof, Hella|Hessmann, Elisabeth|Johnsen, Steven A
PMID: 28369619
Journal: Genome Res. 2017 Nov;27(11):1830-1842.
Title: Altered hydroxymethylation is seen at regulatory regions in pancreatic cancer and regulates oncogenic pathways.
Author: Bhattacharyya, Sanchari|Pradhan, Kith|Campbell, Nathaniel|Mazdo, Jozef|Vasantkumar, Aparna|Maqbool, Shahina|Bhagat, Tushar D|Gupta, Sonal|Suzuki, Masako|Yu, Yiting|Greally, John M|Steidl, Ulrich|Bradner, James|Dawlaty, Meelad|Godley, Lucy|Maitra, Anirban|
PMID: 28986391