Primary Site >> Colorectal Cancer

Gene >> PRMT5

  • 2007
  • 2012
  • 2015
  • 2017
  • 2018
Ref: Inhibition of the heat shock protein 90 molecular chaperone in vitro and in vivo by novel, synthetic, potent resorcinylic pyrazole/isoxazole amide analogues.
PMID: 17431102
Ref: Arginine methylation controls growth regulation by E2F-1.
PMID: 22327218
Ref: Targeting protein arginine methyltransferase 5 inhibits colorectal cancer growth by decreasing arginine methylation of eIF4E and FGFR3.
PMID: 26078354
Ref: High nuclear expression of protein arginine methyltransferase-5 is a potentially useful marker to estimate submucosal invasion in endoscopically resected early colorectal carcinoma.
PMID: 26248553
Ref: Coronin 2A (CRN5) expression is associated with colorectal adenoma-adenocarcinoma sequence and oncogenic signalling.
PMID: 26373535
Ref: Discovery of selective protein arginine methyltransferase 5 inhibitors and biological evaluations.
PMID: 27714957
Ref: Adapting AlphaLISA high throughput screen to discover a novel small-molecule inhibitor targeting protein arginine methyltransferase 5 in pancreatic and colorectal cancers.
PMID: 28591716
Ref: Development of an AlphaLISA high throughput technique to screen for small molecule inhibitors targeting protein arginine methyltransferases.
PMID: 29099132
Ref: Protein arginine methyltransferase 5 is implicated in the aggressiveness of human hepatocellular carcinoma and controls the invasive activity of cancer cells.
PMID: 29749478
Ref: Sirtuin 7-mediated deacetylation of WD repeat domain 77 (WDR77) suppresses cancer cell growth by reducing WDR77/PRMT5 transmethylase complex activity.
PMID: 30282801