Primary Site >> Colorectal Cancer

Gene >> TPI1

Journal: Int J Oncol. 2004 Sep;25(3):571-8.
Title: A novel combination antimetabolite, TAS-102, exhibits antitumor activity in FU-resistant human cancer cells through a mechanism involving FTD incorporation in DNA.
Author: Emura, Tomohiro|Suzuki, Norihiko|Yamaguchi, Masahiro|Ohshimo, Hideyuki|Fukushima, Masakazu
PMID: 15289858
Journal: Anticancer Drugs. 2005 Mar;16(3):285-92.
Title: Determinants of trifluorothymidine sensitivity and metabolism in colon and lung cancer cells.
Author: Temmink, Olaf H|de Bruin, Michiel|Comijn, Elizabeth M|Fukushima, Masakazu|Peters, Godefridus J
PMID: 15711180
Journal: Int J Biochem Cell Biol. 2007;39(3):565-75.
Title: Activity and substrate specificity of pyrimidine phosphorylases and their role in fluoropyrimidine sensitivity in colon cancer cell lines.
Author: Temmink, Olaf H|de Bruin, Michiel|Turksma, Annelies W|Cricca, Silvia|Laan, Adrie C|Peters, Godefridus J
PMID: 17098463
Journal: J Immunol. 2010 Jun 1;184(11):6529-36.
Title: Novel SHP-1 inhibitors tyrosine phosphatase inhibitor-1 and analogs with preclinical anti-tumor activities as tolerated oral agents.
Author: Kundu, Suman|Fan, Keke|Cao, Mingli|Lindner, Daniel J|Zhao, Zhizhaung Joe|Borden, Ernest|Yi, Taolin
PMID: 20421638
Journal: Mol Cancer Ther. 2010 Aug;9(8):2287-96.
Title: Tyrosine phosphatase inhibitor-3 sensitizes melanoma and colon cancer to biotherapeutics and chemotherapeutics.
Author: Kundu, Suman|Fan, Keke|Cao, Mingli|Lindner, Daniel J|Tuthill, Ralph|Liu, Lili|Gerson, Stanton|Borden, Ernest|Yi, Taolin
PMID: 20682647
Journal: Exp Ther Med. 2011 May;2(3):393-397.
Title: Trifluorothymidine exhibits potent antitumor activity via the induction of DNA double-strand breaks.
Author: Suzuki, Norihiko|Nakagawa, Fumio|Nukatsuka, Mamoru|Fukushima, Masakazu
PMID: 22977515
Journal: Br J Cancer. 2012 Jul 24;107(3):429-34.
Title: Phase I study of TAS-102 treatment in Japanese patients with advanced solid tumours.
Author: Doi, T|Ohtsu, A|Yoshino, T|Boku, N|Onozawa, Y|Fukutomi, A|Hironaka, S|Koizumi, W|Sasaki, T
PMID: 22735906
Journal: World J Gastroenterol. 2014 Sep 7;20(33):11840-9.
Title: Identification of differential proteins in colorectal cancer cells treated with caffeic acid phenethyl ester.
Author: He, Yu-Jun|Li, Wan-Ling|Liu, Bao-Hua|Dong, Hui|Mou, Zhi-Rong|Wu, Yu-Zhang
PMID: 25206290
Journal: Oncol Rep. 2014 Dec;32(6):2319-26.
Title: Repeated oral dosing of TAS-102 confers high trifluridine incorporation into DNA and sustained antitumor activity in mouse models.
Author: Tanaka, Nozomu|Sakamoto, Kazuki|Okabe, Hiroyuki|Fujioka, Akio|Yamamura, Keisuke|Nakagawa, Fumio|Nagase, Hideki|Yokogawa, Tatsushi|Oguchi, Kei|Ishida, Keiji|Osada, Akiko|Kazuno, Hiromi|Yamada, Yukari|Matsuo, Kenichi
PMID: 25230742
Journal: Ther Adv Med Oncol. 2015 Nov;7(6):340-56.
Title: Therapeutic potential of TAS-102 in the treatment of gastrointestinal malignancies.
Author: Peters, Godefridus J
PMID: 26557901
Journal: Invest New Drugs. 2015 Oct;33(5):1068-77.
Title: Phase I study of TAS-102 and irinotecan combination therapy in Japanese patients with advanced colorectal cancer.
Author: Doi, Toshihiko|Yoshino, Takayuki|Fuse, Nozomu|Boku, Narikazu|Yamazaki, Kentaro|Koizumi, Wasaburo|Shimada, Ken|Takinishi, Yasutaka|Ohtsu, Atsushi
PMID: 26163340
Journal: Int J Oncol. 2015;46(6):2327-34.
Title: Crucial roles of thymidine kinase 1 and deoxyUTPase in incorporating the antineoplastic nucleosides trifluridine and 2'-deoxy-5-fluorouridine into DNA.
Author: Sakamoto, Kazuki|Yokogawa, Tatsushi|Ueno, Hiroyuki|Oguchi, Kei|Kazuno, Hiromi|Ishida, Keiji|Tanaka, Nozomu|Osada, Akiko|Yamada, Yukari|Okabe, Hiroyuki|Matsuo, Kenichi
PMID: 25901475
Journal: Oncol Rep. 2015 May;33(5):2135-42.
Title: Efficacy of combination chemotherapy using a novel oral chemotherapeutic agent, TAS-102, together with bevacizumab, cetuximab, or panitumumab on human colorectal cancer xenografts.
Author: Tsukihara, Hiroshi|Nakagawa, Fumio|Sakamoto, Kazuki|Ishida, Keiji|Tanaka, Nozomu|Okabe, Hiroyuki|Uchida, Junji|Matsuo, Kenichi|Takechi, Teiji
PMID: 25812794
Journal: Expert Rev Clin Pharmacol. 2016;9(3):355-65.
Title: A novel antimetabolite: TAS-102 for metastatic colorectal cancer.
Author: Miyamoto, Yuji|Lenz, Heinz-Josef|Baba, Hideo
PMID: 26677869
Journal: Anticancer Res. 2016 Jan;36(1):21-6.
Title: TAS-102 an Emerging Oral Fluoropyrimidine.
Author: Chen, Jiezhong|Han, Mei|Saif, Muhammad Wasif
PMID: 26722024
Journal: Clin Cancer Res. 2016 Jun 15;22(12):2835-9.
Title: TAS-102 for Treatment of Advanced Colorectal Cancers That Are No Longer Responding to Other Therapies.
Author: van der Velden, Daphne L|Opdam, Frans L|Voest, Emile E
PMID: 27126991
Journal: Crit Rev Oncol Hematol. 2016 Aug;104:91-7.
Title: Review on TAS-102 development and its use for metastatic colorectal cancer.
Author: Mota, Jose Mauricio|Fonseca, Leonardo G|Braghiroli, Maria Ignez|Hoff, Paulo M
PMID: 27296058
Journal: Am J Cancer Res. 2017 Oct 1;7(10):2032-2040. eCollection 2017.
Title: Synergistic anticancer activity of a novel oral chemotherapeutic agent containing trifluridine and tipiracil in combination with anti-PD-1 blockade in microsatellite stable-type murine colorectal cancer cells.
Author: Suzuki, Norihiko|Tsukihara, Hiroshi|Nakagawa, Fumio|Kobunai, Takashi|Takechi, Teiji
PMID: 29119052
Journal: Am J Cancer Res. 2017 Dec 1;7(12):2577-2586. eCollection 2017.
Title: Combined efficacy and mechanism of trifluridine and SN-38 in a 5-FU-resistant human colorectal cancer cell lines.
Author: Matsuoka, Kazuaki|Takechi, Teiji
PMID: 29312810
Journal: Anticancer Res. 2018 Mar;38(3):1427-1434.
Title: Pre-exposure to Fluorouracil Increased Trifluridine Incorporation and Enhanced its Anti-tumor Effect for Colorectal Cancer.
Author: Baba, Taisuke|Kokuryo, Toshio|Yamaguchi, Junpei|Yokoyama, Yukihiro|Uehara, Keisuke|Ebata, Tomoki|Nagino, Masato
PMID: 29491068
Journal: Oncotarget. 2018 Jan 1;9(26):18559-18569.
Title: Identification of specific and common diagnostic antibody markers for gastrointestinal cancers by SEREX screening using testis cDNA phage library.
Author: Kobayashi, Sohei|Hiwasa, Takaki|Arasawa, Takahiro|Kagaya, Akiko|Ishii, Sayaka|Shimada, Hideaki|Ito, Masaaki|Suzuki, Masae|Kano, Masayuki|Rahmutulla, Bahityar|Kitamura, Kouichi|Sawabe, Yuji|Shin, Hideo|Takiguchi, Masaki|Nomura, Fumio|Matsubara, Hisahiro|Ma
PMID: 29719626
Journal: Clin Colorectal Cancer. 2018 Sep;17(3):e531-e539.
Title: Real-world Treatment Patterns Among Patients With Colorectal Cancer Treated With Trifluridine/Tipiracil and Regorafenib.
Author: Patel, Anuj K|Duh, Mei S|Barghout, Victoria|Yenikomshian, Mihran A|Xiao, Yongling|Wynant, Willy|Tabesh, Majid|Fuchs, Charles S
PMID: 29803544
Journal: J Cell Physiol. 2018 Nov;233(11):8919-8929.
Title: Triose-phosphate isomerase is a novel target of miR-22 and miR-28, with implications in tumorigenesis.
Author: Lone, Saife Niaz|Maqbool, Raihana|Parray, Fazl Q|Ul Hussain, Mahboob
PMID: 29856481
Journal: Int J Mol Sci. 2018 Sep 25;19(10). pii: ijms19102915.
Title: Effective Sequential Combined Chemotherapy with Trifluridine/Tipiracil and Regorafenib in Human Colorectal Cancer Cells.
Author: Matsuoka, Kazuaki|Nakagawa, Fumio|Tanaka, Nozomu|Okabe, Hiroyuki|Matsuo, Kenichi|Takechi, Teiji
PMID: 30257515